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^ See ⇒Homologous competitive binding curves Archived 2007-12-19 at the Wayback Machine., A complete guide to nonlinear regression, curvefit.com.
^ Baaske P, Wienken CJ, Reineck P, Duhr S, Braun D (March 2010). “Optical thermophoresis for quantifying the buffer dependence of aptamer binding”. Angewandte Chemie 49 (12): 2238?41. doi:10.1002/anie.200903998. PMID 20186894 (February 24, 2010).
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^ Matera, Carlo; Flammini, Lisa; Quadri, Marta; Vivo, Valentina; Ballabeni, Vigilio; Holzgrabe, Ulrike; Mohr, Klaus; De Amici, Marco et al. (2014-03-21). “Bis(ammonio)alkane-type agonists of muscarinic acetylcholine receptors: Synthesis, in vitro functional characterization, and in vivo evaluation of their analgesic activity”. European Journal of Medicinal Chemistry 75: 222?232. doi:10.1016/j.ejmech.2014.01.032. PMID 24534538.
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^ Blum JJ, Conn PM (December 1982). “Gonadotropin-releasing hormone stimulation of luteinizing hormone release: A ligand-receptor-effector model”. Proceedings of the National Academy of Sciences of the United States of America 79 (23): 7307?11. Bibcode: 1982PNAS...79.7307B. doi:10.1073/pnas.79.23.7307. JSTOR 13076. PMC 347328. PMID 6296828. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC347328/.
^ Conn PM, Rogers DC, Stewart JM, Niedel J, Sheffield T (April 1982). “Conversion of a gonadotropin-releasing hormone antagonist to an agonist”. Nature 296 (5858): 653?5. Bibcode: 1982Natur.296..653C. doi:10.1038/296653a0. PMID 6280058.
^ Nimczick M, Pemp D, Darras FH, Chen X, Heilmann J, Decker M (August 2014). “Synthesis and biological evaluation of bivalent cannabinoid receptor ligands based on hCB?R selective benzimidazoles reveal unexpected intrinsic properties”. Bioorganic & Medicinal Chemistry 22 (15): 3938?46. doi:10.1016/j.bmc.2014.06.008. PMID 24984935.
^ Russo O, Berthouze M, Giner M, Soulier JL, Rivail L, Sicsic S, Lezoualc'h F, Jockers R, Berque-Bestel I (September 2007). “Synthesis of specific bivalent probes that functionally interact with 5-HT(4) receptor dimers”. Journal of Medicinal Chemistry 50 (18): 4482?92. doi:10.1021/jm070552t. PMID 17676726.
^ Soulier JL, Russo O, Giner M, Rivail L, Berthouze M, Ongeri S, Maigret B, Fischmeister R, Lezoualc'h F, Sicsic S, Berque-Bestel I (October 2005). “Design and synthesis of specific probes for human 5-HT4 receptor dimerization studies”. Journal of Medicinal Chemistry 48 (20): 6220?8. doi:10.1021/jm050234z. PMID 16190749.
^ a b Busnelli M, Kleinau G, Muttenthaler M, Stoev S, Manning M, Bibic L, Howell LA, McCormick PJ, Di Lascio S, Braida D, Sala M, Rovati GE, Bellini T, Chini B (August 2016). “Design and Characterization of Superpotent Bivalent Ligands Targeting Oxytocin Receptor Dimers via a Channel-Like Structure”. Journal of Medicinal Chemistry 59 (15): 7152?66. doi:10.1021/acs.jmedchem.6b00564. PMID 27420737.
^ Lensing CJ, Adank DN, Wilber SL, Freeman KT, Schnell SM, Speth RC, Zarth AT, Haskell-Luevano C (February 2017). “A Direct in Vivo Comparison of the Melanocortin Monovalent Agonist Ac-His-DPhe-Arg-Trp-NH2 versus the Bivalent Agonist Ac-His-DPhe-Arg-Trp-PEDG20-His-DPhe-Arg-Trp-NH2: A Bivalent Advantage”. ACS Chemical Neuroscience 8 (6): 1262?1278. doi:10.1021/acschemneuro.6b00399. PMC 5679024. PMID 28128928. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5679024/.
^ a b Xu L, Josan JS, Vagner J, Caplan MR, Hruby VJ, Mash EA, Lynch RM, Morse DL, Gillies RJ (December 2012). “Heterobivalent ligands target cell-surface receptor combinations in vivo”. Proceedings of the National Academy of Sciences of the United States of America 109 (52): 21295?300. Bibcode: 2012PNAS..10921295X. doi:10.1073/pnas.1211762109. JSTOR 42553664. PMC 3535626. PMID 23236171. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3535626/.
^ a b Lensing CJ, Freeman KT, Schnell SM, Adank DN, Speth RC, Haskell-Luevano C (April 2016). “An in Vitro and in Vivo Investigation of Bivalent Ligands That Display Preferential Binding and Functional Activity for Different Melanocortin Receptor Homodimers”. Journal of Medicinal Chemistry 59 (7): 3112?28. doi:10.1021/acs.jmedchem.5b01894. PMC 5679017. PMID 26959173. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5679017/.
^ Shonberg J, Scammells PJ, Capuano B (June 2011). “Design strategies for bivalent ligands targeting GPCRs”. ChemMedChem 6 (6): 963?74. doi:10.1002/cmdc.201100101. PMID 21520422.
^ Berque-Bestel I, Lezoualc'h F, Jockers R (December 2008). “Bivalent ligands as specific pharmacological tools for G protein-coupled receptor dimers”. Current Drug Discovery Technologies 5 (4): 312?8. doi:10.2174/157016308786733591. PMID 19075611.
^ Akgun E, Javed MI, Lunzer MM, Powers MD, Sham YY, Watanabe Y, Portoghese PS (November 2015). “Inhibition of Inflammatory and Neuropathic Pain by Targeting a Mu Opioid Receptor/Chemokine Receptor5 Heteromer (MOR-CCR5)”. Journal of Medicinal Chemistry 58 (21): 8647?57. doi:10.1021/acs.jmedchem.5b01245. PMC 5055304. PMID 26451468. https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5055304/.

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